Gametocyte clearance kinetics determined by quantitative magnetic fractionation in Melanesian children with uncomplicated malaria treated with artemisinin combination therapy
Journal Title
Antimicrobial Agents and Chemotherapy
Publication Type
Journal Article in press
Abstract
Quantitative magnetic fractionation and a published mathematical model were used to characterize between-treatment differences in gametocyte density and prevalence in 70 Papua New Guinean children with uncomplicated falciparum and/or vivax malaria randomized to one of two artemisinin combination therapies (artemether-lumefantrine or artemisinin-naphthoquine) in an intervention trial. There was an initial rise in peripheral Plasmodium falciparum gametocyte density with both treatments, but it was more pronounced in the artemisinin-naphthoquine group. Model-derived estimates of the median pre-treatment sequestered gametocyte population were 21/muL for artemether-lumefantrine and 61/muL for artemisinin-naphthoquine (P<0.001). The median time for P. falciparum gametocyte density to fall to <2.5/muL (below which transmission becomes unlikely), was 16 days in the artemether-lumefantrine group and 20 days in artemisinin-naphthoquine-treated patients (P<0.001). Gametocyte prevalence modelling suggested that artemisinin-naphthoquine-treated children became gametocytemic faster (median 2.2 days) than artemether-lumefantrine-treated children (5.3 days; P<0.001) and had a longer median P. falciparum gametocyte carriage time per individual (20 vs 13 days; P<0.001). Clearance of P. vivax gametocytes was rapid (within three days) in both groups but, consistent with reappearances of asexual forms in the main trial, nearly 40% of children in the artemether-lumefantrine group developed P. vivax gametocytemia between Days 28 and 42 compared with 3% in artemisinin-naphthoquine-treated children. These data suggest that artemisinin is less active against sequestered gametocytes than artemether. Greater initial gametocyte release after artemisinin-naphthoquine increases the period of potential P. falciparum transmission by four days relative to artemether-lumefantrine but the longer elimination half-life of naphthoquine vs lumefantrine suppresses P. vivax recurrence and consequent gametocytemia.
Publisher
ACS
Research Division(s)
Population Health And Immunity
PubMed ID
25987625
Terms of Use/Rights Notice
Refer to copyright notice on published article.


Creation Date: 2015-05-22 11:19:36
Last Modified: 2019-04-01 09:00:03
An error has occurred. This application may no longer respond until reloaded. Reload 🗙